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Educational purposes only. Not medical advice. Consult healthcare professionals before use.

Healing & Recovery
Preclinical

Brilacidin

Brilacidin

Also known as: PMX-30063, Defensin Mimetic, Host Defense Peptide Mimetic

Overview

Key Facts

Primary Goal: Research and therapeutic applications of Brilacidin

Mimics the amphipathic structure of human beta-defensins. Disrupts bacterial membrane integrity via electrostatic interaction.

Dosing Information

Half-Life

~8 hours

Typical Dose

0.6–1.2 mg

Frequency

1x daily

Cycle Length

7-14 days (acute infection), longer for chronic use

Administration Routes:
oraltopicalintravenous

Benefits

  • Broad-spectrum antimicrobial activity (Gram-positive and Gram-negative bacteria)
  • Anti-biofilm activity against drug-resistant organisms
  • Immunomodulatory effects that enhance host defence
  • Low propensity for bacterial resistance development
  • Anti-inflammatory properties complementing antimicrobial action
  • Potential antiviral activity against enveloped viruses

Side Effects

Infusion-related reactions (IV administration)mild
Nausea (mild to moderate)mild
Headachemild
Localized skin irritation with topical usemild
Transient elevation of liver enzymes (rare)mild

Mechanism of Action

1

Mimics the amphipathic structure of human beta-defensins

2

Disrupts bacterial membrane integrity via electrostatic interaction

3

Inhibits bacterial lipopolysaccharide (LPS) signaling

4

Modulates macrophage and dendritic cell cytokine profiles

5

Resists common bacterial resistance mechanisms (efflux pumps, enzymatic degradation)

Contraindications

Do not use this peptide if any of the following apply:

  • Known hypersensitivity to defensin-mimetic compounds
  • Severe hepatic impairment
  • Pregnancy or breastfeeding
  • Concurrent nephrotoxic agent use (monitor renal function)

Storage & Reconstitution

Unreconstituted (Powder)

Temperature2–8°C (36–46°F)
DurationUp to 3 months

Reconstituted (Mixed)

Temperature2–8°C (36–46°F)
Duration2-4 weeks

Research Summary

Preclinical

Developed by Innovation Pharmaceuticals (formerly Cellceutix). Completed Phase 2 clinical trials for acute bacterial skin and skin structure infections (ABSSSI) with positive results. Also studied for oral mucositis and inflammatory bowel disease. Investigated as potential COVID-19 therapeutic. Represents a novel class of non-peptide immune defence mimetics.

Frequently Asked Questions

Common questions about Brilacidin

UK-Specific Information

Exclusive data points and guidance for UK residents using Brilacidin

UK Lab Testing

UK Lab Testing

Recommended labs: Medichecks, Thriva (£89-£149 for peptide safety panel)

Why this matters: UK-specific lab testing guidance not available on US competitor sites

Commonly Stacked With

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